DEVELOPMENT OF TDPI INHIBITORS BASED ON DERIVATIVES OF CHROMENE AS POTENTIAL ANTI-CANCER DRUGS

A. A Chepanova , N. S Li-Zhulanov , T. A Kurgina , A. L Zakharenko , O. D Zakharova , K. P Volcho , N. F Salakhutdinov , O. I Lavrik

Genes & Cells ›› 2020, Vol. 15 ›› Issue (3S) : 68 -69.

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Genes & Cells ›› 2020, Vol. 15 ›› Issue (3S) :68 -69. DOI: 10.23868/gc122713
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DEVELOPMENT OF TDPI INHIBITORS BASED ON DERIVATIVES OF CHROMENE AS POTENTIAL ANTI-CANCER DRUGS

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A. A Chepanova, N. S Li-Zhulanov, T. A Kurgina, A. L Zakharenko, O. D Zakharova, K. P Volcho, N. F Salakhutdinov, O. I Lavrik. DEVELOPMENT OF TDPI INHIBITORS BASED ON DERIVATIVES OF CHROMENE AS POTENTIAL ANTI-CANCER DRUGS. Genes & Cells, 2020, 15(3S): 68-69 DOI:10.23868/gc122713

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References

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Interthal H et al., The tyrosyl-DNA phosphodiesterase Tdp1 is a member of the phospholipase D superfamily. Proc Natl Acad Sci U S A. 2001;98(21):12009-14.

[2]

Kamaletdinova T et al., The Enigmatic Function of PARP1: From PARylation Activity to PAR Readers. Cells. 2019; 8(12),1625;

[3]

Li-Zhulanov et al., A Novel Class of Tyrosyl-DNA Phosphodiesterase 1 Inhibitors That Contains the Octahydro-2H-chromen-4-ol Scaffold. Molecules, 2018, 23(10), 2468;

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